4-Oxo-2-azetidinecarboxylic acid
| Title | Journal |
|---|---|
| Ring splitting of azetidin-2-ones via radical anions. | Organic & biomolecular chemistry 20121021 |
| An expeditious iodine-catalyzed synthesis of 3-pyrrole-substituted 2-azetidinones. | Molecules (Basel, Switzerland) 20120928 |
| Photoelectron spectra of some antibiotic building blocks: 2-azetidinone and thiazolidine-carboxylic acid. | The journal of physical chemistry. A 20120823 |
| An expeditious route to eight-membered heterocycles by nickel-catalyzed cycloaddition: low-temperature C(sp)2-C(sp)3 bond cleavage. | Angewandte Chemie (International ed. in English) 20120820 |
| Kappa agonist CovX-Bodies. | Bioorganic & medicinal chemistry letters 20120615 |
| Regioselective cycloaddition of 3-azetidinones and 3-oxetanones with alkynes through nickel-catalysed carbon-carbon bond activation. | Chemistry (Weinheim an der Bergstrasse, Germany) 20120319 |
| Synthesis and bioactivities of 2-azetidinone derivatives as cholesterol absorption inhibitors. | Medicinal chemistry (Shariqah (United Arab Emirates)) 20111101 |
| Antibacterial agents and cystic fibrosis: synthesis and antimicrobial evaluation of a series of N-thiomethylazetidinones. | ChemMedChem 20111004 |
| Antiplasmodial and cytotoxicity evaluation of 3-functionalized 2-azetidinone derivatives. | Bioorganic & medicinal chemistry letters 20110801 |
| Synthesis of spirocyclic β-keto-lactams: copper catalyzed process. | Chemical communications (Cambridge, England) 20110507 |
| Synthesis, evaluation and structural studies of antiproliferative tubulin-targeting azetidin-2-ones. | Bioorganic & medicinal chemistry 20110401 |
| Monocyclic β-lactams: new structures for new biological activities. | Current medicinal chemistry 20110101 |
| 2-Azetidinone--a new profile of various pharmacological activities. | European journal of medicinal chemistry 20101201 |
| Synthesis of chlorinated bicyclic C-fused tetrahydrofuro[3,2-c]azetidin-2-ones. | The Journal of organic chemistry 20101105 |
| Ferrier-Petasis rearrangement of 4-(vinyloxy)azetidin-2-ones: an entry to carbapenams and carbacephams. | The Journal of organic chemistry 20101015 |
| T-type calcium channel blockers: spiro-piperidine azetidines and azetidinones-optimization, design and synthesis. | Bioorganic & medicinal chemistry letters 20100801 |
| Azetidinone-isothiazolidinones: stereoselective synthesis and antibacterial evaluation of new monocyclic beta-lactams. | Bioorganic & medicinal chemistry 20100501 |
| Synthesis, in-vitro antimicrobial and cytotoxic studies of novel azetidinone derivatives. | Archiv der Pharmazie 20100401 |
| Suppressed beta-effect of silicon in 3-silylated monocyclic beta-lactams: the role of antiaromaticity. | Organic letters 20091217 |
| Design, synthesis and bioactivity of catechin/epicatechin and 2-azetidinone derived chimeric molecules. | Bioorganic & medicinal chemistry letters 20091215 |
| 2-Azetidinone derivatives: design, synthesis, in vitro anti-microbial, cytotoxic activities and DNA cleavage study. | European journal of medicinal chemistry 20091201 |
| Azetidinones as zinc-binding groups to design selective HDAC8 inhibitors. | ChemMedChem 20091201 |
| Lewis acid-assisted ene cyclization of 2-azetidinone-tethered enals: synthesis of enantiopure carbacepham derivatives. | Chemistry, an Asian journal 20091005 |
| Staudinger ketene-imine cycloaddition, RCM approach to macrocrocyclic bisazetidinones. | The Journal of organic chemistry 20090605 |
| Large ring 1,3-bridged 2-azetidinones: experimental and theoretical studies. | European journal of medicinal chemistry 20090501 |
| 2-Azetidinone derivatives: design, synthesis and evaluation of cholesterol absorption inhibitors. | European journal of medicinal chemistry 20090401 |
| Spiro-piperidine azetidinones as potent TRPV1 antagonists. | Bioorganic & medicinal chemistry letters 20090201 |
| Deeper insight into the mechanism of the reaction of photogenerated metallaketenes and imines. | Journal of the American Chemical Society 20081022 |
| Novel syntheses of azetidines and azetidinones. | Chemical reviews 20080901 |
| 3-Alkenyl-2-azetidinones as fatty acid amide hydrolase inhibitors. | Bioorganic & medicinal chemistry letters 20080715 |
| Total synthesis of (-)-kainic acid via intramolecular Michael addition: a second-generation route. | Organic letters 20080501 |
| Discovery of azetidinone acids as conformationally-constrained dual PPARalpha/gamma agonists. | Bioorganic & medicinal chemistry letters 20080315 |
| New regiocontrolled synthesis of functionalized pyrroles from 2-azetidinone-tethered allenols. | Chemistry (Weinheim an der Bergstrasse, Germany) 20080101 |
| Synthesis and biological activity of N-substituted-3-chloro-2-azetidinones. | Molecules (Basel, Switzerland) 20071112 |
| Synthesis of novel N-(4-ethoxyphenyl) azetidin-2-ones and their oxidative N-deprotection by ceric ammonium nitrate. | Molecules (Basel, Switzerland) 20071025 |
| Synthesis of 3-[4'-(p-chlorophenyl)-thiazol-2'-yl]-2-[(substituted azetidinone/thiazolidinone)-aminomethyl]-6-bromoquinazolin-4-ones as anti-inflammatory agent. | Bioorganic & medicinal chemistry 20070415 |
| Azetidinones as vasopressin V1a antagonists. | Bioorganic & medicinal chemistry 20070301 |
| Indium-mediated selective introduction of a 1,3-butadien-2-yl group at the C4-position in 2-azetidinones and application of 1,3-diene-tethered 2-azetidinones in the Diels-Alder reaction. | Chemistry (Weinheim an der Bergstrasse, Germany) 20070101 |
| A theoretical proposal for the synthesis of carbapenems from 4-(2-propynyl)azetidinones promoted by [W(CO)5] as an alternative to the Ag+-assisted process. | Chemistry (Weinheim an der Bergstrasse, Germany) 20061016 |
| Structures of (S)-(-)-4-oxo-2-azetidinecarboxylic acid and 3-azetidinecarboxylic acid from powder synchrotron diffraction data. | Acta crystallographica. Section B, Structural science 20060801 |
| Synthesis of strained tricyclic beta-lactams by intramolecular [2+2] cycloaddition reactions of 2-azetidinone-tethered enallenols: control of regioselectivity by selective alkene substitution. | Chemistry (Weinheim an der Bergstrasse, Germany) 20060201 |
| The polymer-supported and combinatorial synthesis of beta-lactam compounds: an update. | Mini reviews in medicinal chemistry 20060101 |
| Rabbit small intestine does not contain an annexin II/caveolin 1 complex as a target for 2-azetidinone cholesterol absorption inhibitors. | Biochimica et biophysica acta 20060101 |
| Synthesis of 2-azetidinones from 2-diazo-1, 2-diarylethanones and N-(2-thienylidene)imines as possible antimicrobial agents. | Farmaco (Societa chimica italiana : 1989) 20050901 |
| The indium-mediated selective introduction of allenyl and propargyl groups at the C4-position of 2-azetidinones and the AuCl3-catalyzed cyclization of 4-allenyl-2-azetidinones. | Angewandte Chemie (International ed. in English) 20050311 |
| 3,4-disubstituted azetidinones as selective inhibitors of the cysteine protease cathepsin K. Exploring P3 elements for potency and selectivity. | Bioorganic & medicinal chemistry letters 20050301 |
| Kinetics and mechanism of hydrolysis of N-acyloxymethyl derivatives of azetidin-2-one. | The Journal of organic chemistry 20040514 |
| Examination of the 1,4-disubstituted azetidinone ring system as a template for combretastatin A-4 conformationally restricted analogue design. | Bioorganic & medicinal chemistry letters 20040503 |
| Solid-phase synthesis and SAR of 4-carboxy-2-azetidinone mechanism-based tryptase inhibitors. | Bioorganic & medicinal chemistry letters 20040503 |
| Synthesis of optically pure highly functionalized gamma-lactams via 2-azetidinone-tethered iminophosphoranes. | The Journal of organic chemistry 20040206 |
| Synthesis of antitumor 6-alkylidenepenicillanate sulfones and related 3-alkylidene-2-azetidinones. | Bioorganic & medicinal chemistry letters 20040105 |
| Synthesis and evaluation of N1/C4-substituted beta-lactams as PPE and HLE inhibitors. | Bioorganic & medicinal chemistry 20040102 |
| Synthesis of cryptophycins via an N-acyl-beta-lactam macrolactonization. | The Journal of organic chemistry 20031212 |
| Synthesis of a biotin-tagged photoaffinity probe of 2-azetidinone cholesterol absorption inhibitors. | Bioorganic & medicinal chemistry 20030417 |
| Catalysts with mixed ligands on immobilized supports. Electronic and steric advantages. | Organic letters 20030220 |
| Synthesis and SAR of 4-carboxy-2-azetidinone mechanism-based tryptase inhibitors. | Bioorganic & medicinal chemistry letters 20021104 |
| A stereoselective synthesis of BMS-262084, an azetidinone-based tryptase inhibitor. | The Journal of organic chemistry 20020531 |
| General approach for the stereocontrolled construction of the beta-lactam ring in amino acid-derived 4-alkyl-4-carboxy-2-azetidinones. | The Journal of organic chemistry 20020531 |
| Water-assisted alkaline hydrolysis of monobactams: a theoretical study. | Chemistry (Weinheim an der Bergstrasse, Germany) 20020215 |
| Synthesis of iodinated biochemical tools related to the 2-azetidinone class of cholesterol absorption inhibitors. | Bioorganic & medicinal chemistry letters 20020211 |
| Synthesis of fluorescent biochemical tools related to the 2-azetidinone class of cholesterol absorption inhibitors. | Bioorganic & medicinal chemistry letters 20020211 |
| Design, synthesis and pharmacological evaluation of 3-benzylazetidine-2-one-based human chymase inhibitors. | Bioorganic & medicinal chemistry 20011101 |
| Metal-promoted allylation, propargylation, or allenylation of azetidine-2,3-diones in aqueous and anhydrous media. Application to the asymmetric synthesis of densely functionalized 3-substituted 3-hydroxy-beta-lactams. | The Journal of organic chemistry 20010727 |
| Crystal structure of 3,3-dichloro-N-p-methoxyphenyl-4-(2-phenylstryl)-2-azetidinone. | Analytical sciences : the international journal of the Japan Society for Analytical Chemistry 20010701 |
| Entry to new conformationally constrained amino acids. First synthesis of 3-unsubstituted 4-alkyl-4-carboxy-2-azetidinone derivatives via an intramolecular N(alpha)-C(alpha)-cyclization strategy. | The Journal of organic chemistry 20010518 |
| beta-lactam derivatives as enzyme inhibitors: carboxy peptidyl derivatives of (S)-4-oxoazetidine-2-carboxylate as peptidomimetics. | Archiv der Pharmazie 20010501 |
| Design, synthesis and stability of N-acyloxymethyl- and N-aminocarbonyloxymethyl-2-azetidinones as human leukocyte elastase inhibitors. | Bioorganic & medicinal chemistry letters 20010423 |
| Synthesis of trans-4-aryl-3-(omega-chloroalkyl) -2-azetidinones. | Mededelingen (Rijksuniversiteit te Gent. Fakulteit van de Landbouwkundige en Toegepaste Biologische Wetenschappen) 20010101 |